Cat No.
CEI-1060
Abbr
InSolution? JAK Inhibitor I(Jak1, Jak2, Jak3, Tyk2)
Alias
RP23-336G7.2, AA960307, C130039L05Rik
Synonyms
RP23-336G7.2, AA960307, C130039L05Rik
CAS No.
457081-03-7
IC50
15 nM, 1 nM, 5 nM, 1 nM
Targets
murine JAK1, JAK2, JAK3, Tyk2
Chemical Name
2-(1,1-Dimethylethyl)-9-fluoro-3,6-dihydro-7H-benz[h]-imidaz[4,5-f]isoquinolin-7-one, P6, Pyridone 6, DBI, JAK1 Inhibitor I, JAK2 Inhibitor I, JAK3 Inhibitor X
M.Wt
309.3
Purity
>98% by HPLC
Solubility
A 10 mM (500 μg/162 μl) solution of JAK Inhibitor I (Cat. No. 420099) in DMSO.
Storage
+2 centigrade to +8 centigrade

