Cat No.
CEI-1075
Description
BMS-911543 is a potent and selective inhibitor of JAK2 with IC50 of 1.1?nM, ~350-, 75- and 65-fold selective to JAK1, JAK3 and TYK2, respectively. Phase 1/2.
Abbr
BMS-911543(JAK2)
Alias
JTK10, THCYT3
Synonyms
JTK10, THCYT3
CAS No.
1271022-90-2
IC50
1.1?nM
Targets
JAK2
Chemical Name
Imidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide, N,N-dicyclopropyl-4-[(1,5-dimethyl-1H-pyrazol-3-yl)amino]-6-ethyl-1,6-dihydro-1-methyl-
M.Wt
432.52
Storage
2 years -20 centigrade Powder
2 weeks4centigradein DMSO
6 months-80centigradein DMSO