Cat No.
CEI-1073
Description
CEP33779 is a selective JAK2 inhibitor with IC50 of 1.8 nM, >40- and >800-fold versus JAK1 and TYK2.
Abbr
CEP-33779(JAK2)
Alias
JTK10, THCYT3
Synonyms
JTK10, THCYT3
CAS No.
1257704-57-6
IC50
1.8 nM
Targets
JAK2
Chemical Name
[1,2,4]Triazolo[1,5-a]pyridin-2-amine, N-[3-(4-methyl-1-piperazinyl)phenyl]-8-[4-(methylsulfonyl)phenyl]-
M.Wt
462.57
Purity
0.9918
Solubility
DMSO 93 mg/mL
Water <1 mg/mL
Ethanol <1 mg/mL
Storage
2 years -20 centigrade Powder
2 weeks4centigradein DMSO
6 months-80centigradein DMSO