Cat No.
CEI-1117
Description
TG-46 is a JAK inhibitor.
Abbr
TG-46(JAK2, FLT3, RET, JAK3)
Alias
JTK10, THCYT3
Synonyms
JTK10, THCYT3
CAS No.
936091-15-5
IC50
6nM, 25nM, 17nM, 169nM
Product_Overview
JAK inhibitor
Targets
JAK2, FLT3, RET, JAK3
Chemical Name
N-(1,1-dimethylethyl)-3-[[5-methyl-2-[[4-(4-methyl-1-pipera zinyl)phenyl]amino]-4-pyrimidinyl]amino]-Benzenesulfonamide
M.Wt
510.65
Purity
> 95%
Solubility
DMSO > 112mg/mL Water >1mg/mL Ethanol > 4mg/mL
Storage
4 centigrade
Stability
2 years -20 centigrade Powder
1 month -4 centigrade in DMSO
More than one month -80 centigrade in DMSO