SD-06

 
 
单价 面议对比
询价 暂无
浏览 980
发货 北京
过期 长期有效
更新 2025-05-05 15:00
 

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详细说明
Cat No.
CEI-1107
Description
SD-06 is a p38 MAP kinase inhibitor. It inhibits p38α with an IC50 value of 170nM and inhibits LPS-stimulated TNF-release in rats (83% inhibition at 1mg/kg, po).
Abbr
SD-06(MAPK14)
Alias
RP1-179N16.5, CSBP, CSBP1, CSBP2, CSPB1, EXIP, Mxi2, PRKM14, PRKM15, RK, SAPK2A, p38, P38alpha
Synonyms
RP1-179N16.5, CSBP, CSBP1, CSBP2, CSPB1, EXIP, Mxi2, PRKM14, PRKM15, RK, SAPK2A, p38, P38alpha
CAS No.
271576-80-8
Product_Overview
p38 MAP kinase inhibitor
Targets
MAPK (p38MAP)
Chemical Name
1-(4-(5-(4-chlorophenyl)-4-(pyrimidin-4-yl)-1H-pyrazol-3-yl)piperidin-1-yl)-2-hydroxyethanone
M.Wt
397.86
Purity
> 95%
Solubility
DMSO > 112mg/mL Water >1mg/mL Ethanol > 4mg/mL
Storage
4 centigrade
Stability
2 years -20 centigrade Powder 1 month -4 centigrade in DMSO More than one month -80 centigrade in DMSO
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