AMG-51

 
 
单价 面议对比
询价 暂无
浏览 599
发货 北京
过期 长期有效
更新 2025-05-06 00:13
 

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详细说明
Cat No.
CEI-1119
Description
It shows the enzyme selectivity of c-Met with Ki=4.9nM, KDR with Ki=139nM, Ron with Ki=28nM, IGFR with Ki=22nM.
Abbr
AMG-51(MET)
Alias
AUTS9, HGFR, RCCP2, c-Met
Synonyms
AUTS9, HGFR, RCCP2, c-Met
CAS No.
890019-63-3
Product_Overview
c-Met, KDR, Ron, IGFR inhibitors
Targets
c-Met, KDR, Ron, IGFR
Chemical Name
5-(3-fluoro-4-(6-methoxy-7-(3-morpholinopropoxy)quinolin-4-yloxy)phenyl)-2-(4-fluorophenylamino)-3-methylpyrimidin-4(3H)-one
M.Wt
629.65
Purity
> 95%
Solubility
DMSO > 112mg/mL Water >1mg/mL Ethanol > 4mg/mL
Storage
-20 centigrade
Stability
2 years -20 centigrade Powder 1 month -4 centigrade in DMSO More than one month -80 centigrade in DMSO
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