Cat No.
CEI-0093
Description
Equivalent to the IC50 for wild-type PI3K-alpha, PKI-402 inhibits E545K and H1047R PI3K-alpha mutants with IC50 of 3 nM.
CAS No.
1173204-81-3
Targets
PI3Kalpha
Chemical Name
1-(4-(3-ethyl-7-morpholino-3H-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl)phenyl)-3-(4-(1-methylpiperazine-4-carbonyl)phenyl)urea
M.Wt
570.65
Purity
>99%
Solubility
DMSO 0.4 mg/mL,Water
Storage
2 years at -20 centigrade
