MK 3207 HCl

 
 
单价 面议对比
询价 暂无
浏览 855
发货 北京
过期 长期有效
更新 2026-10-24 00:44
 

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详细说明
Cat No.
CEI-0342
Description
MK 3207 HCl
CAS No.
957116-20-0
Targets
CGRP
M.Wt
594.05
Purity
>99%
Solubility
No
Storage
2 years at -20 centigrade
In vitro
Although has affinity for AMY1 (CTR/RAMP1) receptor with a Ki value of 0.75 nM, MK 3207 displays marked selectivity for human CGRP receptor versus related human AM1 (CLR/RAMP2) receptor, AM2 (CLR/RAMP3) receptor, AMY3 (CTR/RAMP3) receptor, and CTR with Ki values of 16.5 uM, 0.156 uM, 0.128 uM and 1.9 uM, respectively.
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