Cat No.
CEI-1154
Description
PD 0332991 (Palbociclib) Isethionate is the isethionate of PD 0332991, a highly specific inhibitor of CDK4 and CDK6 with IC50 of 11 nM and 16 nM, respectively.
Abbr
PD-0332991 Isethionate(CDK4, CDK6)
Alias
CMM3, PSK-J3
Synonyms
CMM3, PSK-J3
IC50
11 nM, 16 nM
Targets
CDK4, CDK6
Chemical Name
6-acetyl-8-cyclopentyl-5-methyl-2-((5-(piperazin-1-yl)pyridin-2-yl)amino)pyrido[2,3-d]pyrimidin-7(8H)-one
M.Wt
573.66
Purity
> 95%
Storage
4 centigrade