Cat No.
CEI-1146
Description
SAR131675 inhibits VEGFR-3 tyrosine kinase activity with an IC50 20nM and VEGFR-3 autophosphorylation in HEK cells with an IC50 45nM.
Abbr
SAR131675(FLT4)
Alias
FLT41, LMPH1A, PCL, VEGFR3
Synonyms
FLT41, LMPH1A, PCL, VEGFR3
CAS No.
1092539-44-0
Targets
VEGFR-3
Chemical Name
(R)-2-amino-1-ethyl-7-(3-hydroxy-4-methoxy-3-methylbut-1-yn-1-yl)-N-methyl-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxamide
M.Wt
358.39
Purity
> 95%
Storage
4 centigrade