Cat No.
CEI-0596
Description
Cell-permeable. A potent, competitive, and reversible antagonist of the orphan receptor GPR35 (Ki = 12.8 nM). Prevents the GPR35-mediated increase in ERK1/2 phosphorylation and β-arrestin recruitment induced by pamoic acid.
CAS No.
264233-05-8
Product_Overview
A potent and reversible antagonist of the orphan receptor GPR36
Targets
GPR35
Chemical Name
Methyl -5-((2-t-butylcarbamothioyl)hydrazono)methyl)-1-(2,4-difluorophenyl)-1H-pyrazole-4-carboxylate
M.Wt
259.33
Purity
>98% by TLC
Appearance
Yellow solid
Solubility
DMSO (~25 mg/ml) or EtOH (~ 6 mg/ml)
Storage
-20 centigrade
Shipping Conditions
Gel pack
Handling
Protect from air and light
Usage
For Research Use Only! Not For Use in Humans.
