Cat No.
CEI-1168
Description
PF-06405761 is a selective BET (bromodomain-containing protein) inhibitor for BRD4 with IC50 of 0.22 μM.
Abbr
PF-06405761(BRD4)
Alias
CAP, HUNK1, HUNKI, MCAP
Synonyms
CAP, HUNK1, HUNKI, MCAP
CAS No.
1403764-72-6
IC50
0.22 μM
Targets
BRD4
Chemical Name
2-methoxy-N-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-6-yl)benzenesulfonamide
M.Wt
347.39
Purity
> 95%
Storage
4 centigrade