Cat No.
CEI-0342
Description
MK 3207 HCl
CAS No.
957116-20-0
Targets
CGRP
M.Wt
594.05
Purity
>99%
Solubility
No
Storage
2 years at -20 centigrade
In vitro
Although has affinity for AMY1 (CTR/RAMP1) receptor with a Ki value of 0.75 nM, MK 3207 displays marked selectivity for human CGRP receptor versus related human AM1 (CLR/RAMP2) receptor, AM2 (CLR/RAMP3) receptor, AMY3 (CTR/RAMP3) receptor, and CTR with Ki values of 16.5 uM, 0.156 uM, 0.128 uM and 1.9 uM, respectively.