Cat No.
CEI-0974
Description
Selective inhibitor of Ca2+-calmodulin-dependent protein kinase kinase (Ki = 80 and 15 ng/ml for inhibition of CaM-KKalpha and CaM-KKbeta respectively). Binds to the ATP-binding site. Displays >80-fold selectivity over CaMK1, CaMK2, CaMK4, MLCK, PKC, PKA and p42 MAPK. Cell permeable.
Abbr
STO-609(CAMKK2)
Alias
7-oxo-7H-benzimidazo[2, 1-a]benz[de]isoquinoline-3-carboxylic acid acetate
Synonyms
7-oxo-7H-benzimidazo[2,1-a]benz[de]isoquinoline-3-carboxylic acid acetate
CAS No.
52029-86-4
Product_Overview
CAMKK inhibitor
Targets
CAMKK
M.Wt
314.3
Purity
98% (TLC); NMR (Conforms)
Appearance
Yellow powder
Solubility
May be dissolved in: DMSO (10 mg/ml)